Eisner, JR; Abbott, DH; Bird, IM; Rafferty, SW; Moore, WR; Schotzinger, RJ. VT-464: A Novel, Selective Inhibitor of P450c17(CYP17)-17,20 Lyase for Castration-Refractory Prostate Cancer (Poster Presentation) 2012 Genitourinary Cancers Symposium, San Francisco, CA, United States, February 2-4, 2012 (2012).
Pisle, ST; Spencer, SD; Pressler, HM; Troutman, SM; Eisner, JR; Rafferty, SW; Schotzinger, RJ; Moore, WR; Figg, WD. Activity of Oral VT-464, a Selective CYP17 Lyase Inhibitor in the LNCap Prostate Cancer Xenograft (Poster Presentation) 2012 Genitourinary Cancers Symposium, San Francisco, CA, United States, February 2-4, 2012 (2012).
Rafferty, SW; Eisner, JR; Hoekstra, WJ; Higgins, AJ; Schotzinger, R. In-vitro Potency and Safety Index of Three Novel P450c17 17,20-Lyase Inhibitors (Poster Presentation) 92nd Annual ENDO Meeting, San Diego, CA, United States, June 19-22, 2010 (2010).
Norris, John David; Joseph, James David; Sherk, Andrea Barreto; Juzumiene, Dalia; Turnbull, Philip Stewart; Rafferty, Stephen William; Cui, Huaxia; Anderson, Erin; Fan, Daju; Dye, Delita Arnelle; et al Differential Presentation of Protein Interaction Surfaces on the Androgen Receptor Defines the Pharmacological Actions of Bound Ligands Chemistry & Biology (Cambridge, MA, United States) (2009), 16(4), 452-460.
Rafferty, Stephen. From selective PPAR ligands to PPAR pan-agonists. Oral Presentation (Invited Speaker) Advancing the Efficacy, Safety and Selectivity of Metabolic Disease Therapeutics, Chapel Hill, NC, March 17 - 19, 2008.
Rafferty, Stephen; Gampe, Robert; Han, Bajin; Randhawa, Sab A.; Stewart, Eugene L.; Yates, Christopher M. Benzoxazepinones: The discovery of a novel SARM template. Abstracts of Papers, 234th ACS National Meeting, Boston, MA, United States, August 19-23, 2007 (2007).
Guo, Jiasheng; Erickson, Greg A.; Fitzgerald, Russ N.; Matsuoka, Richard T.; Rafferty, Stephen W.; Sharp, Matthew J.; Sickles, Barry R.; Wisowaty, James C. An Efficient Synthesis of a Potent PPARpan Agonist. Journal of Organic Chemistry (2006), 71(21), 8302-8305.
Rafferty, Stephen; Banker, Pierette; Henke, Brad R.; Lambert, Millard H.; Oliver, William; Sternbach, Daniel D. From selective PPAR ligands to PPAR pan-agonists. Oral Presentation, 230th ACS National Meeting, Washington, DC, United States, Aug. 28-Sept. 1, 2005.
Rafferty, Stephen; Wisowaty, James; Matsuoka, Richard; Martin, Michael; Guo, Jiasheng. Highly regioselective addition of thiophenols to 2-(4-trifluoromethylphenyl)-4,5-bis(hydroxymethyl)thiazoles in the synthesis of PPAR agonists. Poster Presentation, 224th ACS National Meeting, Boston, MA, United States, August 18-22, 2002.
Presentation: The Discovery of Potent and Selective PPAR-alpha agonists
Authors: Stephen W. Rafferty, Peter J. Brown, Rodolfo Cadilla
Meeting: Glaxo-Wellcome International Chemistry Meeting (GWICM) in Verona, Italy
Date: April, 1999.
Crimmins, Michael T.; Rafferty, Stephen W. Regioselective and stereoselective reductive cleavage of 1,7-dioxaspiro[5.5]undecane alcohols. Tetrahedron Letters (1996), 37(32), 5649-5652.
Rafferty, Stephen W. The Regio- and Stereoselective Reductive Cleavage of Spiroketals, Oral Presentation, ACS North Carolina Section Meeting, Raleigh, North Carolina, April 1995.